PD 173212

>99%

N-type Ca2+ channels

Synthetic

PD 173212 (#P-105) is a highly pure, synthetic, and biologically active compound.

599.9

PD 173212 is a dipeptidyl-amine that acts as an N-type voltage-gated Ca2+ channel blocker1. PD 173212 inhibited N-type channels in IMR-32 cells with IC50 = 36 nM as measured by Ca2+ imaging of K+ stimulated cells and only had small effects on other channels at much higher concentrations1.

DMSO. Centrifuge all product preparations before use (10000 x g 5 min).

10 nM - 10 μM.

Lyophilized

C38H53N3O3.

217171-01-2

Up to four weeks at 4°C or three months at -20°C.