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Arachidonyl serotonin

品牌： Absin

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参数

分子式：

C₃₀H₄₂N₂O₂

分子量：

462.7

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产品介绍

产品信息

商品描述

N-Arachidonoyl-serotonin is a selective FAAH (fatty acid amid hydrolase) and VR1 (transient receptor potential vanilloid-1, TRPV1) channel inhibitor. TRPV1 is a Capsaicin receptor, which behaves as a non-selective cation channel and are mainly found in the sensory neurons that detect painful stimuli. The compound has been shown to be inactive against cPLA2 and CB1. Rat brain studies suggests that N-Arachidonoyl-serotonin acts as an enhancer of endocannabinoid levels, and increases the levels of anadamide and 2-AG .

分子量

462.7

纯度

98%

可溶性

Soluble in DMSO (>25 mg/mL), ethanol (15 mg/mL), DMF (30 mg/mL), and PBS (pH 7.2) (~290 µg/mL).

外观

Oil

IC50

fatty acid amide hydrolase (FAAH): IC₅₀ = 5.6 mM; TRPV1: IC₅₀ = 40 nM

应用

实验应用

A selective FAAH and TRPV1 channel inhibitor

背景

分子式

C₃₀H₄₂N₂O₂

CAS号

187947-37-1

沸点

680.49° C at 760 mmHg (Predicted)

MDL

MFCD02179189

PK值

pK_a: 10.08 (Predicted)

密度

1.04 g/mL (Predicted)

折射率

n²⁰_D 1.57 (Predicted)

制备和贮存

保存方式

Store at -20° C

参考图片

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货号：

abs42022970-10mg

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